Friday, July 08, 2011

Maraviroc Abacavir STudy - Effect on Endothelial Recovery

HIV infected patients treated with abacavir might have a higher risk for the occurrence of cardiovascular events. At time of writing of this protocol the underlying mechanism is not yet elucidated, however some studies find impaired endothelial function and elevated markers of chronic inflammation in these patients,suggesting a higher lever of chronic inflammation. Recently maraviroc...

Brief Summary

Official Title: “Maraviroc Abacavir STudy - Effect on Endothelial Recovery”

HIV infected patients treated with abacavir might have a higher risk for the occurrence of cardiovascular events. At time of writing of this protocol the underlying mechanism is not yet elucidated, however some studies find impaired endothelial function and elevated markers of chronic inflammation in these patients,suggesting a higher lever of chronic inflammation.

Recently maraviroc (Celsentri®), a CCR5-receptor antagonist, became available for treatment of patients infected with HIV-1.

Improvement of endothelial function may be a potential beneficial side effect of treatment with maraviroc, due to the potential reduction of immune activation and chronic inflammation as a result of blocking the CCR5-coreceptor. Moreover, treatment intensification of HAART with maraviroc in patients with suppressed plasma HIV_RNA may decrease plasma HIVRNA below the cut-off of 50 copies/ml as well.

The investigators hypothesize that maraviroc intensification therapy in patients on an abacavir-containing regimen will improve endothelial function.

The objectives of this study are: First, to assess the effect of addition of maraviroc to an abacavir-containing regimen on endothelial function; second, to assess the effect of this intervention on markers of immune activation and chronic inflammation, and on plasma HIV-RNA below 50 copies/ml.


  • Study Type: Interventional


  • Study Design: Allocation: Randomized, Endpoint Classification: Efficacy Study, Intervention Model: Crossover Assignment, Masking: Open Label, Primary Purpose: Treatment


  • Study Primary Completion Date: September 2012



  • Detailed Clinical Trial Description

    The MASTER study is a phase IV, randomized, open label, cross-over, intervention study.

    Study subjects who are on stable abacavir-containing regimen will be randomized into two arms. In arm A maraviroc will be added to their regimen at baseline, while study subjects in arm B will continue their abacavir-containing regimen. After 8 weeks, cross-over of the study arms will be performed. Subjects in arm A will then stop maraviroc, while in subjects in arm B maraviroc will be added to their regimen (for 8 weeks again). The total duration of the study will be 16 weeks.

    Intervention(s) in this Clinical Trial

    Drug: Maraviroc
    HAART of subjects enrolled in arm A will be intensified with maraviroc during week 1-8.

    Arms, Groups and Cohorts in this Clinical Trial

    Active Comparator: Arm A
    HAART of subjects in arm A will be intensified with maraviroc during week 1-8.
    Active Comparator: Arm B
    HAART of subjects enrolled in arm B will be intensified with maraviroc during week 9-16
    Outcome Measures for this Clinical Trial

    Primary Measures

    Change in flow-mediated dilatation (FMD) of the brachial artery after 8 weeks of maraviroc treatment as compared to the control group
    Time Frame: After 8 weeks of treatment (cross-over)
    Safety Issue?: No

    Secondary Measures

    Change in markers of chronic inflammation
    Time Frame: Baseline, week 2 (A) or 10 (B), week 4 (A) or 12 (B), week 8, week 16
    Safety Issue?: No
    Change in markers of immune activation
    Time Frame: Baseline, week 2 (A) or 10 (B), week 4 (A) or 12 (B), week 8, week 16
    Safety Issue?: No
    Change in markers of endothelial function
    Time Frame: Baseline, week 2 (A) or 10 (B), week 4 (A) or 12 (B), week 8, week 16
    Safety Issue?: No
    Changes in plasma HIV-RNA below 50 copies/ml
    Time Frame: Baseline, week 8, week 16
    Safety Issue?: No
    Change in endothelial function measured by EndoPAT
    Time Frame: baseline, week 8, week 16
    Safety Issue?: No

    Criteria for Participation in this Clinical Trial

    Inclusion Criteria:

    Age > 18 years
    HIV-1 infection
    Treatment with antiretroviral regimen containing abacavir for at least the previous 3 months
    Undetectable plasma HIV RNA (50 cp/ml) for at least 6 months (one 'blip' allowed, which is defined as a detectable plasma HIV-RNA level between 50 and 400 copies/ml, preceded and followed by undetectable (<50 copies/ml) plasma HIV-RNA measurements) CD4+ cell count > 200 cells/µL
    Signed informed consent

    Exclusion Criteria:

    Pregnancy
    Breastfeeding
    Allergy for peanuts or soya
    Hypersensitivity for maraviroc
    Treatment of underlying malignancy
    Acute infection in the preceding 30 days
    Renal insufficiency requiring hemodialysis
    Acute or decompensated chronic hepatitis
    Modification of antiretroviral regimen in the previous 3 months
    Gender Eligibility for this Clinical Trial: Both

    Minimum Age for this Clinical Trial: 18 Years

    Maximum Age for this Clinical Trial: N/A

    Are Healthy Volunteers Accepted for this Clinical Trial?: No

    Clinical Trial Investigator Information

    Lead Investigator: UMC Utrecht Other

    Overall Clinical Trial Officials and Contacts

    A IM Hoepelman, MD, PhD Principal Investigator UMC Utrecht

    Overall Contact: Steven FL van Lelyveld, MD s.f.l.vanlelyveld@umcutrecht.nl

    Additional Information

    Information obtained from ClinicalTrials.gov on July 06, 2011
    Link to the current ClinicalTrials.gov record. http://clinicaltrials.gov/show/NCT01389063
    Study ID Number: MASTER2010
    ClinicalTrials.gov Identifier: NCT01389063
    Health Authority: Netherlands: The Central Committee on Research Involving Human Subjects (CCMO)

    Copyright © 2011 ClinicalTrials

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